PhI(OAc)2/I2 induced aziridination of alkenes with TsNH2 under mild conditions |
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Authors: | Renhua Fan Dongming Pu Bing Wang |
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Affiliation: | a Department of Chemistry, Fudan University, 220 Handan Road, Shanghai 200433, China b College of Food Science, Shanghai Fisheries University, 334 Jungong Road, Shanghai 200090, China |
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Abstract: | The aziridination of alkenes with the direct use of p-toluenesulfonamide (TsNH2) was achieved by using PhI(OAc)2 and I2 under mild conditions. The reaction affords aziridines in moderate to good yields, and offers good manipulability by avoiding the use of the expensive metal catalyst and the unstable and explosive PhINTs. |
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