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Disruptor of telomeric silencing 1-like (DOT1L): disclosing a new class of non-nucleoside inhibitors by means of ligand-based and structure-based approaches
Authors:Manuela Sabatino  Dante Rotili  Alexandros Patsilinakos  Mariantonietta Forgione  Daniela Tomaselli  Fréderic Alby  Paola B. Arimondo  Antonello Mai  Rino Ragno
Affiliation:1.Rome Center for Molecular Design, Dipartimento di Chimica e Tecnologie del Farmaco,Sapienza Università di Roma,Roma,Italy;2.Dipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur - Fondazione Cenci Bolognetti,Sapienza Università di Roma,Roma,Italy;3.Alchemical Dynamics s.r.l.,Roma,Italy;4.Laboratoire Pierre Fabre,Toulouse,France;5.CNRS FRE3600 ETaC, Bat IBCG,Toulouse,France;6.Oversea Fellow, Churchill College,Cambridge,UK
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