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Virtual Ligand Screening of the p300/CBP Histone Acetyltransferase: Identification of a Selective Small Molecule Inhibitor
Authors:Erin M Bowers  Gai Yan  Chandrani Mukherjee  Andrew Orry  Ling Wang  Marc A Holbert  Nicholas T Crump  Catherine A Hazzalin  Glen Liszczak  Hua Yuan  Cecilia Larocca  S Adrian Saldanha  Ruben Abagyan  Yan Sun  David J Meyers  Ronen Marmorstein  Louis C Mahadevan  Rhoda M Alani  Philip A Cole
Institution:1. Department of Pharmacology and Molecular Sciences, Johns Hopkins University School of Medicine, Baltimore, MD 21205, USA;2. Department of Oncology, Johns Hopkins University School of Medicine, Baltimore, MD 21205, USA;3. Molsoft LLC, La Jolla, CA 92037, USA;4. Nuclear Signalling Laboratory, Department of Biochemistry, Oxford University, Oxford OX1 3QU, UK;5. Program in Gene Expression and Regulation, The Wistar Institute, Philadelphia, PA 19104, USA;6. The Scripps Research Institute, Jupiter, FL 33458, USA;7. Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California, San Diego, La Jolla, CA, 92093, USA;8. Department of Chemistry, University of Pennsylvania, Philadelphia, PA 19104, USA
Abstract:
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