排序方式: 共有32条查询结果,搜索用时 15 毫秒
1.
Siddiqui Madiha M. Nagargoje Amol A. Akolkar Satish V. Sangshetti Jaiprakash N. Khedkar Vijay M. Pisal Parshuram M. Shingate Bapurao B. 《Research on Chemical Intermediates》2022,48(3):1199-1225
Research on Chemical Intermediates - A simple and efficient protocol has been developed for the synthesis of new1,2,3-triazole-2,3-dihydroquinazolin-4[1H]-one (DHQ) conjugates(6a?j) via... 相似文献
2.
Danne Ashruba B. Choudhari Amit S. Sarkar Dhiman Sangshetti Jaiprakash N. Khedkar Vijay M. Shingate Bapurao B. 《Research on Chemical Intermediates》2018,44(10):6283-6310
Research on Chemical Intermediates - The synthesis of a new series of triazole-biscoumarin conjugates by using a molecular hybridization approach is described. The newly synthesized compounds... 相似文献
3.
Jaiprakash N. Sangshetti Nagnnath D. Kokare Sandeep A. Kotharkar Devanand B. Shinde 《Monatshefte für Chemie / Chemical Monthly》2008,139(2):125-127
Summary. 2,4,5-Triaryl-1H-imidazoles were efficiently synthesized from benzoin or benzil, ammonium acetate, and aromatic or heteroaromatic aldehydes
in the presence of sodium bisulfite as catalyst. The present protocol offers significant improvements for the synthesis of
2,4,5-triaryl-1H-imidazoles with regard to yield of products, simplicity in operation, and cheap catalyst. 相似文献
4.
Jaiprakash N. Sangshetti Devanand B. Shinde Nagnnath D. Kokare 《Journal of heterocyclic chemistry》2008,45(4):1191-1194
5.
A simple,efficient,and environment benign route was developed for the preparation of bis-(indolyl)methanes and 14-aryl-14H-dibenzo[a,j]xanthenes from condensation of various aromatic aldehydes or ketones with indole,and 2-naphthol,respectively,using oxalic acid catalyst in aqueous medium.Use of cheap and easily available catalyst,better yields and simple reaction protocol are the advantages of the present method. 相似文献
6.
Jaiprakash N. Sangshetti Nagnnath D. Kokare Devanand B. Shinde 《中国化学快报》2007,18(11):1305-1308
Sulfanilic acid has been found to be an efficient catalyst for the synthesis of 1,5-benzodiazepines from o-phenylenediamine and ketones. This method is simple, effective and environmentally friendly and gives better yields. 相似文献
7.
Nagnnath D. Kokare Jaiprkash N. Sangshetti Devanand B. Shinde 《中国化学快报》2007,18(11):1309-1312
Oxalic acid was found to be an efficient catalyst for Pechmann condensation,which includes the reaction between phenols andβ-keto esters leading to formation of coumarin derivatives.The advantages of present methods are the use of cheap and easy available catalyst,solvent-free reaction conditions,better yields and shorter reaction time. 相似文献
8.
Jaiprakash N. Sangshetti Nagnnath D. Kokare Sandeep A. Kotharkar Devanand B. Shinde 《Monatshefte für Chemie / Chemical Monthly》2008,7(3):125-127
2,4,5-Triaryl-1H-imidazoles were efficiently synthesized from benzoin or benzil, ammonium acetate, and aromatic or heteroaromatic aldehydes
in the presence of sodium bisulfite as catalyst. The present protocol offers significant improvements for the synthesis of
2,4,5-triaryl-1H-imidazoles with regard to yield of products, simplicity in operation, and cheap catalyst. 相似文献
9.
Zahid Zaheer Firoz A. Kalam Khan Jaiprakash N. Sangshetti Rajendra H. Patil 《中国化学快报》2016,27(2):287-294
A series of novel 3-substituted-4-hydroxycoumarin derivatives 6(a–1) were synthesized in high yield using one-pot three component coupling reaction catalyzed by ceric ammonium nitrate. These compounds were evaluated for antileishmanial activity against Leishmania donovani promastigotes and antioxidant activity(DPPH-radical scavenging activity). Two compounds, 6h(IC_(50)= 9.90 μmol/L) and 6i(IC_(50)= 6.90 μmol/L) displayed potent antileishmanial activity when compared with standard antileishmanial agents pentamidine(IC_(50)= 16.15 μmol/L) and miltefosine(IC_(50)= 12.50 μmol/L). Three compounds, 6c(IC_(50)= 10.79 μmol/L), 6h(IC50= 10.60 μmol/L), and 6i(IC_(50)= 10.73 μmol/L) showed significant antioxidant activity favorably with the antioxidant standards butylated hydroxy toluene(IC_(50)= 16.47 μmol/L) and ascorbic acid(IC_(50)= 12.69 μmol/L). A molecular docking study of compounds 6(a–1) suggested a possible mode of binding with the Adenine phosphoribosyltransferase enzyme of L.donovani. ADME properties were predicted in silico and support the potential of 6(a–1) to show favorable drug-like properties. 相似文献
10.
ZrOCl2·8H2O catalyzed environmentally benign synthesis of isobenzofuran-1(3H)-ones are described.ZrOCl2·8H2O appeared to be an excellent catalyst for the condensation and reactions.Reaction of phthalaldehydic acid(2-carboxybenzaldehyde) with methylaryl and cyclic ketones was initiated by condensation and occurred in one step providing excellent yields(90-98%). 相似文献