Arylhydroxyacetic acids and amino acids derived from ethinylphenols

Conclusions A method of synthesis of arylhydroxyacetic acids and ammo acids derived from ethinylphenols has been developed in view of possible physiological activity of these compounds.Translated from Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, No. 5, pp. 1170–1172, May, 1970.     

Alkynyl derivatives of benzofuran

A general method for the preparation of alkynyl derivatives of benzofuran, including -ethynylbenzofuran, consists in the cyclization of o-mono-and dialkynylphenols under the conditions of the Mannich and Cadiot-Chodkiewicz reactions.Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 11, pp. 1457–1460, November, 1972.     

Synthesis and study of antimicrobial action of amino derivatives of 4-hydroxy-4′-ethynylazobenzene

Conclusions In order to manifest bacteriological activity in the series of the morpholine and piperdine derivatives of ethynylazobenzene it is important to have present a free hydroxyl group and only one triple bond in the molecule.Translated from Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, No. 4, pp. 978–980, April, 1972.     

Acetylenic derivatives of aniline

Conclusions The direct condensation of iodoanilines with 2-methyl-3-bu1yn-2-ol gave acetylenic carbinols, whose cleavage by the reverse Favorskii reaction leads to ethynylanilines.Translated from Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, No. 5, pp. 1184–1186, May, 1982.     

Diacetylene alcohol derivatives of aromatic amines

Conclusions We have developed methods of synthesis of acetylenic and diacetylenic alcohol derivatives of simple aromatic amines.Translated from Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, No. 4, pp. 821–823, April, 1984.