资讯

刘延东强调:充分发挥科学技术的引领支撑作用中共中央政治局委员、国务委员刘延东在全国科技工作会议上强调,科技系统要深刻认识党中央、国务院明确把科技放在优先发展地位的重大战略意义,自觉肩负起历史使命,紧密结合新形势新任务,深入贯彻落实科学发展观,加强自主创新,加快科技成果的转化应     

用声音给手机充电

这可能是史上又一个令人尴尬的发明——日前,韩国科学家发明了一种装置,可以让手机在通话时利用声音进行充电。该技术可将声音转化为电能,用户在打电话的时候手机就会进行充电,而且是声音越大,充电越快。这对于爱煲电话粥的人来说,简直是天大的喜讯,但也许未来会有许多人在公共场合为了给手机充电而大声喧哗。     

高职学生顶岗实习——让学校与企业无缝对接

本文根据指导高职学生顶岗实习的工作经历,阐述了高职学生顶岗实习对学校和对企业的积极意义。     

一种简便、有效的水蒸汽蒸馏装置在半微量有机实验中的应用

分析了一种简便、有效的水蒸汽蒸馏装置在半微量有机实验中的应用。该装置具有节约能源、占实验台面积小、安装拆卸方便、整个实验完成时间短等优点。     

电气化铁路接触网除冰装置

本期新开栏目“发明达人秀”，是一个专门为小发明家及科技爱好者开办的栏目，无论您的作品是否获奖，只要是原创发明都可以拿到我们的秀场show出来。每期由读者评出一个发明小擂主，每期擂主将获得参加年度评选的参赛资格，年末由读者及专家评选出“年度达人”，可获得本刊为您提供的精美奖品及证书。欢迎大家踊跃采稿!     

通信传输业务对接问题分析

本文就通信传输对接问题常见故障现象及其原因、故障定位思路和方法进行阐述,通过分析典型案例,加深对对接问题处理的理解,提高了处理传输业务对接故障的能力。     

国际资讯

英国首测太阳能垃圾桶近日,英国开始太阳能垃圾桶的首次试验,这种新式垃圾桶可以利用太阳能对垃圾进行压缩,其容量是普通垃圾桶的8倍,堪称垃圾桶中的大胃王。这项试验一旦成功,将带来新一轮的环保技术革命。这种新式垃圾桶只需要少量的阳光就可实现对垃圾的压缩,垃圾桶中装有一个传感器,在负重达到一定程度时,会     

Asymmetric Synthesis, Antifungal Activity and Molecular Modeling of Iodiconazole Isomers

Iodiconazole is a novel antifungal agent that was developed in its racemic form. In order to investigate the ef- fects of the chiral center on the antifungal activity, R- and S-isomers of iodiconazole were prepared on the basis of the asymmetric Sharpless epoxidation. （S）-Iodiconazole was proved to have better antifungal activity than the （R）- isomer. The binding modes of the two isomers with lanosterol 14~z-demethylase were clarified by molecular dock- ing.     

Triazole and Benzotriazole Derivatives as Novel Inhibitors for p90 Ribosomal S6 Protein Kinase 2： Synthesis, Molecular Docking and SAR Analysis

A series of triazole and benzotriazole derivatives as novel p90 ribosomal S6 protein kinase 2 （RSK2） inhibitors were designed and synthesized. The in vitro activities against RSK2 were evaluated, and among 14 compounds, compounds 5, 6, 11, 12, 13 and 14 exhibited enzyme IC50 values of 8.91, 2.86, 3.19, 3.05, 4.49 and 2.09 μmol/L re- spectively. The proposed binding modes were simulated using molecular docking method, and the docking results coupled with the stmcture-activi1：y relationship （SAR） analysis indicated that all these active compounds bound to the RSK2 ATP binding site at NTKD, and the electron-donating groups on the 4-position of phenyl were the deter- minant point for the inhibitory activity.     

一种改进的汽车尾气检测装置的过滤清洁阀

公开号:CN202691221U公开日:2013.01.23申请人:骆旭山,陶元本实用新型公开了一种改进的汽车尾气检测装置的过滤清洁阀,包括连接于一体的内接口、阀体和外接口,