Synthesis of 5,6-Dihydro-OSW-1 and Its Antitumor Activities

5,6-Dihydro-OSW-1 (1) was synthesized following our previous procedure for the total synthesis of OSW-1. This compound demonstrated slightly stronger potency than that of OSW-1 against the growth of cancer cells.     

Microwave Synthesis, Characterization and DNA-binding Properties of a New Cobalt（ Ⅱ ） Complex with 2,6-Bis（benzimidazol-2-yl）pyridine

A new cobalt(Ⅱ) complex with tridentate ligand 2, 6-bis (benzimidazol-2-yl)pyridine has been synthesized by microwave irradiation method and characterized by elemental analysis,electrochemical and spectral methods. The binding of the complex with calf thymus DNA has also been investigated by absorption and fluorescence spectra.     

One-pot Synthesis of 2, 5-Disubstituted Oxazoles Using Poly[styrene（iodosodiacetate）]

2,5-Disubstituted oxazoles were prepared conveniently by treatment of aromatic α-methyl ketones and nitriles with poly[styrene(iodosodiacetate)] in one-pot process.     

Novel Chiral Ferrocenyl Aziridino Alcohol Catalysts Promoting Asymmetric Addition of Diethylzinc to Aldehydes

Optically active aziridino alcohols containing ferrocenyl groups were prepared from commercially available L-threonine in excellent yields and used as catalysts to promote the asymmetric addition of diethylzinc to aryaldehydes to afford 1-arylpropanol in up to 84% enantiomeric excesses with moderate to good yields.     

例说通过联想类比开发数学问题

创新教育如何体现在教学上 ,对于一个具体的数学问题 ,不妨把它看作一件产品 ,进行联想类比 ;它有哪些变异 ?它还有哪些应用 ?能否开发出更有价值的系列产品 ?下面举例说明进行数学问题这方面的探讨和研究 ,以献读者 . 已知ａ >ｂ>0 ,求ａ+1 6ｂ(ａ-ｂ) 的最小值 ; 已知ａ>ｂ>0 ,求ａ2 +1 6ｂ(ａ -ｂ) 的最小值 (数学第二册上Ｐ37)这是大家熟悉的两个问题 ,通过改造、一般化 ,可得如下结果 :改 1为 :已知ｘ1 ,ｘ2 >0 ,求ｘ1 +ｘ2 +ｋｘ1 ｘ2(ｋ>0且ｋ常数 )的最小值 .解　因ｘ1 ,ｘ2 >0 ,故ｘ1 +ｘ2 +ｋｘ1 ｘ2 ≥3·3 ｋ ,当且仅当ｘ1 =ｘ…     

2003年普通高等学校招生全国统一考试数学（理工农医类）（北京卷）

参考公式与文科相同一 选择题 :本大题共 1 0小题 ,每小题 5分 ,共 5 0分 .在每小题给出的四个选项中 ,只有一项是符合题目要求的 .( 1 ) ,( 2 )与文科 ( 1 ) ,( 2 )相同( 3)“cos2α=- 32 ”是“α=kπ+ 5π1 2 ,k∈Z”的(A)必要非充分条件(B)充分非必要条件(C)充分必要条件(D)既非充分又非必要条件( 4 )与文科 ( 4 )相同( 5 )极坐标方程 ρ2 cos2θ- 2 ρcosθ =1表示的曲线是(A)圆 (B)椭圆(C)抛物线 (D)双曲线( 6) ,( 7) ,( 8)分别与文科 ( 6) ,( 7) ,( 9)相同( 9)若数列 {an}的通项公式是an =3-n+ 2 -n+ ( - 1 ) n( 3-n- 2 -n)2 ,n…     

匹配问题实例空间和解空间结构

本文通过研究匹配问题的实例空间，匈牙利算法和解空间三者之间的关系，指出S实例空间的数目与问题复杂度之间的关系既不是充分也不是必要的，而如何对问题的解空间进行合理的分解才能是问题的关键。     

利用多普勒信息的波达方向最大似然估计方法

为了充分利用信号的时域特性来改善信号波达方向（ＤＯＡ）的估计性能，本文从最大似然估计出发，推导出了有限快拍，低信噪比情况下多普勒信号波达方向的迭代估计计算法，为进一步减小运算量，本文还推导了一种简化算法，本文提出的两种算法对低信噪比，少快拍数下多普勒信号的ＤＯＡ估计性能比不利用时域特性的ＭＬ方法有明显改善，Ｍｏｎｔｅ－Ｃａｒｌｏ实验验证了本文方法的有效性。     

THE RELATIONSHIP BETWEEN PROJECTIVE GEOMETRIC AND RATIONAL QUADRATIC B-SPLINE CURVES

For two rational quadratic B-spline curves with same control vertexes, the cross ratio of four eollinear points are represented; which are any one of the vertexes, and the two points that the ray initialing from the vertex intersects with the corresponding segments of the twocurves, and the point the ray intersecting with the connecting line between the two neighboring vertexes. Different from rational quadratic Beeier curves, the value is generally related with the loeation of the ray, and the necessary and sufficient condition o5 the ratio being independent of the ray‘s loeation is showed. Alsn another cross ratio o5 the following four collinear points are suggested, i.e. one vertex, the points that the ray from the initlal vertex intersects respectivdy with the curve segmentt the line connecting the segments end points, and the line connecting the two neighboring vertexes. This cross ratio is concerned only whh the ray‘s location, butnot with the weights of the curve. Furthermore, the cross ratio is projective invariant under the projective transformation between the two segments.     

A Fixed Point Theorem for Multi—valued Composite Increasing Operators

Ａ　Ｆｉｘｅｄ　Ｐｏｉｎｔ　Ｔｈｅｏｒｅｍ　ｆｏｒ　Ｍｕｌｔｉ－ｖａｌｕｅｄ　Ｃｏｍｐｏｓｉｔｅ　Ｉｎｃｒｅａｓｉｎｇ　ＯｐｅｒａｔｏｒｓＬｉＦｅｎｇｙｏｕ（李凤友）（ＤｅｐａｒｔｍｅｎｔｏｆＭａｔｈｅｍａｔｉｃｓ，Ｔｉａｎｊｉｎ＇ＮｏｒｍａｌＵｎｉ...