A potent and highly selective sulfotransferase inhibitor

In the present work, we have used a newly developed, fluorescence-based assay to screen a library of >30 000 compounds as potential beta-arylsulfotransferase-IV inhibitors. A total of 11 inhibitors were discovered. Most of the compounds discovered showed low micromolar inhibition, but one of the compounds showed potent inhibition (Ki = 96 nM). The most potent of these inhibitors was tested against a variety of other purine binding enzymes and showed remarkable specificity.     

Synthesis of conducting polyaniline using novel anionic Gemini surfactant as micellar stabilizer

The Gemini surfactant 9B-4-9B containing sodium sulfonate as hydrophilic head group was synthesized based on nonylphenol and characterized by FTIR, ¹H NMR spectroscopy and the surface tension measurement. The CMC and C₂₀ of the 9B-4-9B were smaller than that of sodium dodecylbenzene sulfonate and sodium dodecylsulfate, respectively, indicating excellent efficiency of micelle formation and reduced surface tension. Conducting polyaniline salts were synthesized by chemical oxidative micellar polymerization of aniline in water firstly using Gemini surfactant 9B-4-9B as the micelle stabilizer and ammonium peroxydisulfate as the oxidant at 0 °C. The stable polyaniline dispersions have been obtained when the molar ratio of the 9B-4-9B to aniline was equal to or above 0.5 used in the polymerization system. The obtained granular polyaniline particles with the size of 1-2 μm were characterized by FTIR, UV-Vis, SEM, WAXD and conductivity measurement.     

东海北部拖虾渔业的现状与设立拖虾休渔期的建议

本文根据近１０年来拖虾调查和虾类资源动态监测资料，分析了拖虾渔业发展的现状和存在问题，并根据虾类资源种类多，分布区域性明显，主要种类的渔场渔期不同，繁殖期、幼虾的时空分布不同等特点，提出设立拖虾休渔期的建议方案。     

对虾塘综合养殖的模式与原理

对对虾塘综合养殖作了详细论述。根据养殖特点将其归纳成五种典型模式，并从理论上对各种养殖模式的原理及其经济、社会和生态效益作了分析。对对虾塘综合养殖的前景作了展望，并指出了今后研究的方向。     

建设社会主义新农村传媒需要实现"三个转变"

目前中国正在进行的建设社会主义新农村运动,对大众传媒来说,是机遇也是挑战。为了适应建设社会主义新农村的需要,现有的传媒格局、经营观念、新闻报道理念乃至报道方法都要做出相应调整。媒体只有从重视生产报道转向重视生活报道,从重视经济视角报道转向社会视角报道,从媒体精英意识转向平民意识,自觉实现“三个转变”,才能充分发挥传媒报道在新农村建设中的作用。     

太湖地区稻田氮素平衡及其环境效应的研究

应用15N微区试验对氮肥在水稻不同生长期的去向进行研究,结果表明,水稻对氮肥的吸收利用随着作物生长的进行而逐渐提高,氮肥的损失和土壤的残留则逐渐下降.土壤残留的肥料氮主要集中在0～20cm的耕层土壤中,占全部土壤残留肥料氮的85%以上.氮肥的总损失在30.4%～54.4%之间,其中氨挥发损失为25.4%～33.3%,为稻田氮素的最主要损失途径.     

低压电力网标准时间传递研究

结合扩频通信技术原理,给出了一种基于低压电力线网的标准时间传递方案,并讨论了它的网络节点地址分配。该方案结构简单,特别适用于单变压器供电区域内标准时间的传递和分配。     

土壤地下点源入渗的基本特性研究

基于大量的大田土壤点源入渗试验，提出了地下点源入渗系统的新理念——管道-土壤系统，分析了地下点源入渗中累积入渗量与入渗率随时间的变化过程及入渗界面问题，建立了地下点源土壤入渗模型，并利用数理统计理论证明了该模型的有效性。研究成果对研究土壤水分运动理论和指导农业地下灌溉实践都具有重要的意义。     

受损托圈承载能力的有限元计算和分析

综合运用计算机仿真、动力学、有限元分析理论和测试技术等科学理论,并以大型的有限元分析软件ANSYS作为仿真和分析的工具,详细研究不同工况下受损托圈的强度,同时校核了受损托圈的承载能力。