Synthesis, Structure and Biological Activities of Novel Triazole Compounds Containing N,N-Dialkyldithiocarbamate Moiety

Introduction As an important type of fungicides, triazole compounds are highly efficient, low poisonous and inward absorbent.1-3 At present, the studies on triazole derivatives are mainly concentrated on compounds with triazole as the only active group. The report of triazole compounds that contain both triazole group and other active group in a single molecule has rarely been found. Dialkyl-substituted dithiocarbamate salts have also shown interesting biological effects.4 N,N-Dialkyldithio-…     

Investigations on Preparation,Crystal Structure and Thermal Stability of Bis(O-ethylcarbonodithiolato-S,S′)(1,10-phenanthroline-N~1,N~(10))cobalt(II) Complex:[Co(Et-XA)_2·phen]·H_2O (XA=xanthate)

IntroductionTheincreasingcommercialvalueoftransitionmetalcomplexesofxanthateshasarousedconsiderableinterestintheirchemistry .Whiletheiranalyticalapplicationsarewellknown ,1theyarenowfindingextensiveuseinvulcan izationofrubber ,frothfloatationprocessforconcentrationofsulphideores ,asantioxidants ,lubricants ,2 ,3andhavebeenfoundtopossessfungicidalandinsecticidalactivi ties .4 Recently ,molecularrecognitionbetweenhostandguestmolecules ,inclusionphenomenaandnoncovalentmolecularinteractionarefunda…     

Synthesis and Crystal Structure of 2-Chloromethyl-1H-benzimidazole Nitrate, [ClCH_2(C_7H_6N_2)]NO_3

1 INTRODUCTION Benzimidazole is an interesting heterocyclic compound because it is found in various naturally occurring drugs, such as omeprazole, astemizole and emedastine difumarate[1]. The efficacy of sub- stituted benzimidazoles in the treatment of parasitic infections is well known[2～4]. Substituted benzimid- azole moieties are established pharmacophores in parasitic chemotherapy. Bis(2-benzimidazole) and some substituted bis(benzimidazol-2-yl)alkanes have attracted much interest …     

Synthesis and Properties of Polyetherketones Containing Sulfide and Phthalazinone

High molecular weight copoly(ether ketone)s (PEK) based on 4-(4-hydroxyphenyl)-1-phthalazinone (DHPZ)/4,4′-thiobisphenol (TBP)/4,4′-diflourodiphenylketone (DFK) were prepared by nucleophilic substitution polycondensation. The copolymers were characterized by FT- and ^1H-NMR. Thermal properties and solubility of copolymers were studied.     

RZ-DPSK传输系统相位噪声的比较分析

建立了单信道40Gbit／s归零-差分相移键控码（RZ-DPSK）传输系统模型，详细地分析并比较了线性相位噪声和非线性相位噪声对系统性能的影响。结果表明，由放大器自发辐射（ASE）噪声带来的线性相位噪声对传输系统的性能影响最大，ASE与自相位调制（SPM）相互作用引起的Gordon-Mollenauer（G-M）相移次之，带内四波混频（IFWM）的影响最小。在最优输入功率的条件下，由ASE带来的线性相位噪声引起的系统差分相位Q值代价大于204dB，由G-M相移引起的系统差分相位Q值代价小于7．5dB。仿真结果表明，对于采用掺铒光纤放大器（EDFA）级联放大的单信道40Gbit／s RZ-DPSK传输系统，ASE噪声是限制系统无中继传输距离的最主要因素。     

基于海天线提取和混合灰度差的船舶检测方法

为了快速、准确检测海天背景下远距离水平观测的船舶目标,提出了一种基于海天线提取和混合灰度差的船舶检测方法.首先,利用边缘检测算法将图像分为天空、海天线和海面三个区域,并根据海天区域连接点,采用直线拟合方法确定海天线的直线参数;然后提取海天线区域作为目标感兴趣区域,并在去除海面杂波和噪声等干扰后利用混合灰度差水平投影和垂...     

Rutin Inhibits Ox-LDL-Mediated Macrophage Inflammation and Foam Cell Formation by Inducing Autophagy and Modulating PI3K/ATK Signaling

Atherosclerosis (AS) is one of the leading causes of death among the elderly, and is primarily caused by foam cell generation and macrophage inflammation. Rutin is an anti-inflammatory, anti-oxidant, anti-allergic, and antiviral flavonoid molecule, known to have anti-atherosclerotic and autophagy-inducing properties, but its biological mechanism remains poorly understood. In this study, we uncovered that rutin could suppress the generation of inflammatory factors and reactive oxygen species (ROS) in ox-LDL-induced M2 macrophages and enhance their polarization. Moreover, rutin could decrease foam cell production, as shown by oil red O staining. In addition, rutin could increase the number of autophagosomes and the LC3II/I ratio, while lowering p62 expression. Furthermore, rutin could significantly inhibit the PI3K/ATK signaling pathway. In summary, rutin inhibits ox-LDL-mediated macrophage inflammation and foam cell formation by inducing autophagy and modulating PI3K/ATK signaling, showing potential in treating atherosclerosis.     

Load Balancing Routing Algorithm Based on Extended Link States in LEO Constellation Network

As an important part of satellite communication network, LEO satellite constellation network is one of the hot research directions. Since the nonuniform distribution of terrestrial services may cause inter-satellite link congestion, improving network load balancing performance has become one of the key issues that need to be solved for routing algorithms in LEO network. Therefore, by expanding the range of available paths and combining the congestion avoidance mechanism, a load balancing routing...     

Energy Efficiency Analysis of MISO-OFDM Communication Systems Considering Power and Capacity Constraints

In this paper, the energy efficiency of multi-input single-output and orthogonal frequency division multiplexing (MISO-OFDM) communication systems with power and capacity constraints is investigated. By formulating the power allocation problem of MISO-OFDM communication systems, the minimum subchannel transmission power is analyzed with power and capacity constraints. Simulation results indicate that there exists a specific minimum subchannel capacity threshold. Moreover, the energy efficiency of MISO-OFDM communication systems starts to increase only when the minimum subchannel capacity exceeds the specific threshold.     

基于PZT陶瓷谐振技术的光纤相位调制器研究

分析影响了基于压电陶瓷谐振换能器的光纤相位调节的主要参数,并根据参数研制出一种满足性能要求的压电陶瓷光纤相位调制器.结果表明,光纤伸长位移量与光纤直径、压电常数、工作电压及陶瓷直径有关,与压电陶瓷的厚度无关;压电陶瓷光纤相位调制器的具有工作频率高(100 kHz以上),驱动电压低(2～3 V),电容小,介电损耗小,自滤波谐振等特点.