| 含七氟异丙基的氯虫酰胺类似物的设计合成及生物活性 |
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| 引用本文： | 冯启,刘智力,王明忠,熊丽霞,于淑晶,李正名. 含七氟异丙基的氯虫酰胺类似物的设计合成及生物活性[J]. 高等学校化学学报, 2011, 32(1): 74-78 |
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| 作者姓名： | 冯启 刘智力 王明忠 熊丽霞 于淑晶 李正名 |
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| 作者单位： | 南开大学元素有机化学国家重点实验室, 元素有机化学研究所, 天津 300071 |
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| 基金项目： | 国家“九七三”计划项目(批准号:2010CB126106); 国家自然科学基金(批准号:20872069)资助 |
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| 摘 要： | 以氯虫酰胺和氟虫酰胺结构为基础，通过活性基团拼接法，设计合成了一系列新的含七氟异丙基的氯虫酰胺类似物，所有化合物通过了核磁共振氢谱和高分辨质谱的表征，并测试了它们的杀虫和杀菌活性。
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| 关 键 词： | 氯虫酰胺 氟虫酰胺 七氟异丙基 杀虫活性 杀菌活性 |
| 收稿时间： | 2010-03-22 |
Design, Synthesis and Biological Activities of Novel Analogues of Chlorantraniliprole Containing Heptafluoroisopropyl Group |
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| FENG Qi,LIU Zhi-Li,WANG Ming-Zhong,XIONG Li-Xia,YU Shu-Jing,LI Zheng-Ming. Design, Synthesis and Biological Activities of Novel Analogues of Chlorantraniliprole Containing Heptafluoroisopropyl Group[J]. Chemical Research In Chinese Universities, 2011, 32(1): 74-78 |
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| Authors: | FENG Qi LIU Zhi-Li WANG Ming-Zhong XIONG Li-Xia YU Shu-Jing LI Zheng-Ming |
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| Affiliation: | State Key Laboratory of Elemento-Organic Chemistry, Institute of Elemento-Organic Chemistry, Nankai University, Tianjin 300071, China |
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| Abstract: | In order to find novel insecticides targeting the ryanodine receptor with high activity,a series of novel analogues of chlorantraniliprole containing heptafluoroisopropyl group,developed from the structures of chlorantranili-prole and flubendiamide,was designed and synthesized according to the substructure link principle.Their structures were characterized by 1H NMR and HRMS.Their evaluated insecticidal activities show that the introduction of the heptafluoroisopropyl group decreases the activitiy sharply.A... |
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| Keywords: | Chlorantraniliprole Flubendiamide Heptafluoroisopropyl group Insecticidal activity Fungicidal activity |
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