|
|||||
|
|
Short Synthesis of Enantiopure Thieno[2,3‐f]triazolo[1,5‐a][1,4]diazepines and Thieno[2,3‐f][1,4]diazepin‐5‐ones |
|
| Authors: | Giorgio Molteni |
| Affiliation: | Dipartimento di Chimica, Università degli Studi di Milano, Milan, Italy |
| Abstract: | Starting from 2‐carboxy‐3‐thenylazide 1 and enantiopure amines 2 as the chiral building blocks, we developed a two‐step synthesis of the title compounds involving an intramolecular azide cycloaddition as the key step. |
| Keywords: | |