Efficient construction of fused indolines with a 2-quaternary center via an intramolecular Heck reaction with a low catalyst loading |
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| Authors: | Zhao Lei Li Ziyuan Chang Lin Xu Jinyi Yao Hequan Wu Xiaoming |
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| Institution: | State Key Laboratory of Natural Medicines and Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. |
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| Abstract: | An efficient construction of fused indolines with a 2-quaternary center through a palladium-catalyzed intramolecular Heck reaction of N-(2(2-halobenzoxyl)-2,3-disubstituted indoles is disclosed. This protocol provided a straightforward access to diverse fused indolines with good functional group tolerance. |
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