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Solid Phase Synthesis of 3‐Toluenesulfonylglutarimides |
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| Authors: | Meng‐Yang Chang Kuo‐Ging Lin Shui‐Tein Chen Nein‐Chen Chang |
| Abstract: | A novel route for the synthesis of 3‐toluenesulfonylglutarimides on a solid support is described. The cyclization step involves stepwise 3+3] strategy of Rink Amide resin bound onto an α‐toluenesulfonyl group with various α,β‐unsaturated esters. |
| Keywords: | Solid‐phase reaction Stepwise [3+3] strategy Rink Amide resin Glutarimides Thalidomide |