Synthesis of fused heterocycles with a benzazepinone moiety via intramolecular Heck coupling |
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| Authors: | Lionel Joucla |
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| Affiliation: | Laboratoire de Chimie Organique 1, UMR-CNRS 5181, Université Claude Bernard-Lyon 1, Bâtiment 308 CPE Lyon, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne cedex, France |
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| Abstract: | The preparation of fused heterocycles with a benzazepinone moiety was realised via an intramolecular Heck coupling reaction either at position 2 or at position 3 of the heterocyclic system. This method allowed the synthesis of the pyrrolo[2,3-c]azepinone core and Paullone derivatives. |
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| Keywords: | Benzazepinone Palladium Heck Cyclisation |
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