Three-component one-pot synthesis of 1,2,3,4-tetrahydroquinoline derivatives in hexafluoroisopropanol |
| |
| Authors: | Jie Zhou Bai Ling Xu |
| |
| Affiliation: | Institute of Materia. Medica, Chinese Academy of Medical Sciences & Peking Union Medical College, Belting 100050, China |
| |
| Abstract: | The one-pot aza-Diels-Alder reaction of substituted aromatic amines, ethyl glyoxylate and benzyl vinylcarbamate or N-benzyloxycarbonyl 2-pyrroline was conducted in hexafluoroisopropanol, providing the desired 1,2,3,4-tetrahydroquinline derivatives in moderate yields. |
| |
| Keywords: | Aza-Diels-Alder reaction Tetrahydroquinoline Hexafluoroisopropanol (HFIP) Fluorinated solvent |
| 本文献已被 维普 万方数据 ScienceDirect 等数据库收录！ |
| 点击此处可从《中国化学快报》浏览原始摘要信息 |
|
点击此处可从《中国化学快报》下载全文 |
|
