A highly regioselective synthesis of 2-aryl-6-chlorobenzothiazoles employing microwave-promoted Suzuki-Miyaura coupling reaction |
| |
| Authors: | Yeon Heo |
| |
| Institution: | Bioorganic Science Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea |
| |
| Abstract: | Suzuki-Miyaura coupling reactions of 2,6-dichlorobenzothiazole with arylboronic acids, promoted by microwave heating, efficiently produce 2-aryl-6-chlorobenzothiazoles in a highly regioselective manner. This process serves as the foundation for a simple method to rapidly construct 2-aryl-6-chlorobenzothiazole libraries. |
| |
| Keywords: | Suzuki-Miyaura reaction Palladium Boronic acid Microwave Benzothiazole Amination |
| 本文献已被 ScienceDirect 等数据库收录！ |
