PIDA-mediated synthesis of oxazoles through oxidative cycloisomerization of propargylamides |
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| Authors: | Akio Saito |
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| Institution: | Laboratory of Organic Reaction Chemistry, Showa Pharmaceutical University, 3-3165 Higashi-tamagawagakuen, Machida, Tokyo 194-8543, Japan |
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| Abstract: | PIDA phenyliodine(III) diacetate] in AcOH or AcOH-HFIP (hexafluoroisopropanol) efficiently promotes the formation of 2,5-disubstituted oxazoles via the oxidative cycloisomerization of propargylamide derivatives. |
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