| Solvent-and Catalyst-free Synthesis and Antifungal Activities of α-Aminophosphonate Containing Cyclopropane Moiety |
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| 基金项目： | Supported by the National Basic Research Program of China(No.2010B12606). |
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| 摘 要： | Nine new α-aminophosphonate derivatives containing cyclopropane moiety have been synthesized via conventional and microwave irradiation methods under solvent-and catalyst-free condition. The structures of the title compounds have been confirmed by 1H NMR, 31P NMR, FTIR, EI-MS and FTICR-MS. Their antifungal activities were evaluated in vivo and some of the compounds were found to exhibit excellent antifungal activities against Corynespora cassiicola, Pseudomonas syringae pv. Lachrymans, Pseudoperonospora cubensis and Sclerotinia sclerotiorum.
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| 收稿时间： | 2009-05-19 |
Solvent- and Catalyst-free Synthesis and Antifungal Activities of α-Aminophosphonate Containing Cyclopropane Moiety |
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| PAN Li,LIU Xing-hai,SHI Yan-xia,WANG Bao-lei,WANG Su-hua,LI Bao-ju,.... Solvent- and Catalyst-free Synthesis and Antifungal Activities of α-Aminophosphonate Containing Cyclopropane Moiety[J]. Chemical Research in Chinese University, 2010, 26(3): 389-393 |
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| Authors: | PAN Li LIU Xing-hai SHI Yan-xia WANG Bao-lei WANG Su-hua LI Bao-ju ... |
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| Affiliation: | 1. State Key Laboratory of Elemento-Organic Chemistry, National Pesticidal Engineering Centre(Tianjin), Tianjin Key Laboratory of Pesticide Science, Nankai University, Tianjin 300071, P. R. China;
2. Institute of Vegetables and Flowers, Chinese Academy of Agricultural Sciences, Beijing 100081, P. R. China |
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| Abstract: | Nine new α-aminophosphonate derivatives containing cyclopropane moiety have been synthesized via conventional and microwave irradiation methods under solvent- and catalyst-free condition. The structures of the title compounds have been confirmed by 1H NMR, 31P NMR, FTIR, EI-MS and FTICR-MS. Their antifungal activities were evaluated in vivo and some of the compounds were found to exhibit excellent antifungal activities against Corynespora cassiicola, Pseudomonas syringae pv. Lachrymans, Pseudoperonospora cubensis and Sclerotinia sclerotiorum. |
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| Keywords: | α-Aminophosphonate Imine Antifungal activity, |
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