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Copper‐Catalyzed Amidation of Primary and Secondary Alkyl Boronic Esters |
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| Authors: | Dr. Luis M. Mori‐Quiroz Kirk W. Shimkin Dr. Sina Rezazadeh Ryan A. Kozlowski Prof. Dr. Donald A. Watson |
| Affiliation: | Department of Chemistry and Biochemistry, University of Delaware, Newark, DE, USA |
| Abstract: | The oxidative copper‐catalyzed cross‐coupling of functionalized alkyl boronic esters with primary amides is reported. Through the identification of appropriate diketimine ligands, conditions for efficient coupling of both primary and secondary alkyl boronic esters with diverse primary amides, including acetamide, have been developed. |
| Keywords: | alkyl boronic esters amides copper cross-coupling NacNac ligand |