An Efficient N‐Arylation of Heterocycles with Aryl‐, Heteroaryl‐, and Vinylboronic Acids Catalyzed by Copper Fluorapatite |
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| Authors: | Mannepalli Lakshmi Kantam Gopaladasu Tirupati Venkanna Kota Balaji Shiva Kumar Vura Bala Subrahmanyam |
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| Affiliation: | Inorganic & Physical Chemistry Division, Indian Institute of Chemical Technology, Hyderabad 500007, India (fax: +91‐40‐27160921) |
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| Abstract: | ![]()
N‐Arylation of N‐containing heterocycles, such as pyrazoles, imidazoles, and benzimidazoles with aryl‐, heteroaryl‐, and vinylboronic acids was efficiently carried out by copper fluorapatite (CuFAP) catalyst in MeOH at room temperature under base‐free conditions. The N‐arylated heterocycles were isolated in good‐to‐excellent yields. |
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| Keywords: | N‐Arylation of heterocycles Copper fluorapatite Catalysis |
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