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The Lipophilicity Behavior of Three Catechol‐O‐methyltransferase (COMT) Inhibitors and Simple Analogues
Authors:Laura Novaroli  Geraldine Bouchard&#x;Doulakas  Marianne Reist  Barbara Rolando  Roberta Fruttero  Alberto Gasco  Pierre‐Alain Carrupt
Institution:Laura Novaroli,Geraldine Bouchard Doulakas,Marianne Reist,Barbara Rolando,Roberta Fruttero,Alberto Gasco,Pierre‐Alain Carrupt
Abstract:
Keywords:COMT Inhibitors  Parkinson's disease  Pharmacokinetic profiling  Lipophilicity  Blood‐‐brain‐barrier passive permeation  Inhibitors
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