Design,Synthesis, and Biological Evaluation of an Allosteric Inhibitor of HSET that Targets Cancer Cells with Supernumerary Centrosomes |
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Authors: | Ciorsdaidh  A. Watts,Frances  M. Richards,Andreas Bender,Peter  J. Bond,Oliver Korb,Oliver Kern,Michelle Riddick,Paul Owen,Rebecca  M. Myers,Jordan Raff,Fanni Gergely,Duncan  I. Jodrell,Steven  V. Ley |
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Affiliation: | 1. Department of Chemistry, University of Cambridge, Lensfield Road, Cambridge CB2 1EW, UK;2. Cancer Research UK Cambridge Institute, University of Cambridge, Li Ka Shing Centre, Robinson Way, Cambridge CB2 ORE, UK;3. Unilever Centre for Molecular Science Informatics, Department of Chemistry, University of Cambridge, Lensfield Road, Cambridge 1EW, UK;4. Cambridge Crystallographic Data Centre, 12 Union Road, Cambridge CB2 1EZ, UK;5. Cancer Research Technology, Ltd., Babraham Research Campus, Cambridge CB2 3AT, UK;6. Cancer Research Technology, Ltd., Wolfson Institute of Biomedical Research, The Cruciform Building, London WC1E 6BT, UK;7. Sir William Dunn School of Pathology, University of Oxford, South Parks Road, Oxford OX1 3RE, UK |
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